3种熊果苷的研究进展

doi:10.13218/j.cnki.csdc.2015.09.011

Abstract

Abstract: The preparation method,mechanism of whitening action,as well as the application status and the product stability of three kinds of arbutin were summarized and compared.The new product types and new technologies such as liposomes,microemulsions and clathrates were put forward for providing orientation for development of new applications in the future.

Key words: α-arbutin, β-arbutin, deoxyarbutin, whitening, freckle removal

CLC Number:

TQ658

LIU Cai-yun, WU Pei-cheng, LIANG Gao-wei, LUO Xin-ru, ZHOU Dan-man. Progress in development of three kinds of arbutin product[J].China Surfactant Detergent & Cosmetics, 2015, 45(9): 529-532.

References

[1] HAMED S H.Efficacy and mechanism of action of a new tyrosinase inhibitory agent [D].Cincinnati,OH,USA:University of Cincinnati,2004.
[2] INOMATA S,YKOYAMA M,SETO S,et al.High-yield production of arbutin from hydroquinone in suspension culture of Catharanthus roseus plant cell[J].Appl Microbial Biotechol,1991,36(3):315-319.
[3] 赵明强,丁家宜,刘峻,等.人参毛状根生物合成熊果苷的研究[J].中国中药杂志,2001,26(12):819-822.
[4] 宗飞,姚小武,王海滨.β-熊果苷的合成[J].浙江化工,2013,44(8):10-14.
[5] KITAO S,SHIMAOKA Y,SEKINE H.Manufacture of phenyl glycisides with sucrose phosphorylase:JP,06153976 [P].1994-06-03.
[6] 刘春巧,张淑荣,张鹏.嗜麦芽黄单胞菌BT-112催化制备α-熊果苷[J].日用化学工业,2005,35(6):364-383.
[7] 韦祎,张淑荣,刘春巧,等.添加表面活性剂对α-熊果苷发酵的影响[J].化工学报,2007,58(9):2352-2356.
[8] 李晓娇,刘忆明.α-熊果苷合成研究进展[J].保山学院学报,2014,3(2):18-21.
[9] LI LINGJUN,ZHU LIZHI,ZHANG XINYING,et al.Convenient tetrahydropyranylation of alcohols and phenols by catalytic ferric sulfate hydrate (Fe₂(SO₄)₃·xH₂O)[J].Canadian Journal of Chemistry,2005,83(8):1120-1123.
[10] CHOPA A B,SILBESTRI G F,LOCKHART M T.Strategies for the synthesis of bi- and triarylic materials starting from commercially available phenols[J].Journal of Organometallic Chemistry,2005,690(17):3865-3877.
[11] BANDGAR B P,UPPALLA L S,SADAVARTE V S,et al.Facile and selective deprotection of aryl acetates using sodium perborate under mild and neutral condition[J].New J Chem,2002,26(10):1273-1276.
[12] 张文征. 脱氧熊果苷的合成研究[D].杭州:浙江大学,2010.
[13] FUNAYAMA M,ARAKAWA H,YAMAMOTO R,et al.Effects of alpha- and beta- arbutin on activity of tyrosinases from mushroom and mouse melanoma[J].Biosci Biotechnol Biochem,1995,59(1):143-144.
[14] 刘有停. α-熊果苷美白动力学机制及其配伍性和稳定性的研究[D].北京:北京化工大学,2012.
[15] 樊邦棣,刘建贞.熊果苷的生产开发及其应用前景[J].化学化工,1999(3):9-12.
[16] BOISSY R E,VISSCHER M,DELONG M A.D-Arbutin:a novel reversible tyrosinase inhibitor with effective in vivo skin lightening potency[J].Exp Dermatol,2005,14(8):601-608.
[17] CHAWLA S.Effect of deoxyarbutin and its second-generatioin derivatives on melanocyte viability and function [D].Cincinnati,OH,USA:University of Cincinnati,2006.
[18] HWANG J H,LEE B M.Inhibitory effects of plant extracts on tyrosinase,L-DOPA oxidation,and Melanin synthesis[J].J Toxicol Environ Health:Part A,2007,70(5):393-407.
[19] CHAWLA S,KVALNES K,DELONG M A,et al.Deoxyarbutin and its derivatives inhibit tyrosinase activity and melanin synthesis without inducing reactive oxygen species or apoptosis[J].J Drugs Dermatol,2012,11(10):28-34.
[20] 房军,杨艳伟,张伟,等.化妆品中β-熊果苷稳定性研究[J].卫生研究,2009,38(2):214-215.
[21] 佟文鑫,李佳兴,刘东红.化妆品基础环境对β-熊果苷稳定性的影响[J].日用化学品科学,2010,33(11):15-18.
[22] 艾克蕙,梁今明,曾春莲,等.红外光谱法测定祛斑膏霜中熊果苷的含量和稳定性[J].日用化学工业,1999(2):45-47.
[23] YANG C H,CHEN Y S,LAI J S,et al.Determination of the thermodegradation of deoxyarbutin in aqueous solution by high performance liquid chromatography[J].Int J Mol Sci,2010,11(10):3977-3987.
[24] LIN C C,YANG C H,CHANG N F,et al.Study on the stability of deoxyarbutin in an anhydrous emulsion system[J].Int J Mol Sci,2011,12(9):5946-5954.
[25] YANG C H,CHANG N F,CHEN Y S,et al.Comparative study on the photostability of arbutin and deoxyarbutin:Sensitivity to ultraviolet radiation and enhanced photostability by the water-soluble sunscreen,benzophenone-4[J].Biosci Biotechnol Biochem,2013,77(5):1127-1130.
[26] 赖超. 醋氯芬酸醇质体凝胶的研究[D].重庆:重庆医科大学,2012.
[27] MASINI V,BONTE F,MEYBECK A,et al.Cutaneous bioavailability in hairless rats of tretinoin in liposomes or gel[J].Pharm Sci,1993,82(1):17-21.
[28] WEN A H,CHOI M K,KIM D D.Formulation of liposome for topical delivery of arbutin[J].Arch Pharm Res,2006,29(12):1187-1192.
[29] 吴培诚,彭学东.熊果苷柔性脂质体经皮渗透体系的初步研究[J].临床医学工程,2009,16(8):8-10.

Progress in development of three kinds of arbutin product

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